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DERIVATIVES
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PharmDr. Ondřej Holas Ph.D.
Academic staff at Faculty of Pharmacy in Hradec Králové
2 classes
53 publications
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class
Physical Principles of Dosage Forms
+1
GAPS308 |
Faculty of Pharmacy in Hradec Králové
Publications
publication
3 beta-Isoobeticholic acid efficiently activates the farnesoid X receptor (FXR) due to its epimerization to 3 alpha-epimer by hepatic metabolism
2020 |
Faculty of Pharmacy in Hradec Králové, Faculty of Medicine in Hradec Králové, Faculty of Science
publication
Branched PLGA derivatives with tailored drug delivery properties
2020 |
Faculty of Pharmacy in Hradec Králové
publication
Synthesis of Novel Pyrazinamide Derivatives Based on 3-Chloropyrazine-2-carboxamide and Their Antimicrobial Evaluation
2017 |
Faculty of Pharmacy in Hradec Králové
publication
Novel tacrine/acridine anticholinesterase inhibitors with piperazine and thiourea linkers
2014 |
Faculty of Pharmacy in Hradec Králové
publication
Planar Ni(II) 1,2-dithiolenes involving tridentate P-donor ligands
2012 |
Faculty of Pharmacy in Hradec Králové
publication
Synthesis and in vitro evaluation of 7-methoxy-N-(pent-4-enyl)-1,2,3,4-tetrahydroacridin-9-amine - new tacrine derivate with cholinergic properties
2011 |
Faculty of Pharmacy in Hradec Králové, Faculty of Physical Education and Sport, First Faculty of Medicine
publication
Pseudo-catalytic scavenging: Searching for a suitable reactivator of phosphorylated butyrylcholinesterase
2010 |
Central Library of Charles University
publication
Synthesis and in vitro evaluation of new tacrine derivatives - bis-alkylene linked 7-MEOTA
2010 |
Central Library of Charles University
publication
Evaluation of novel reactivators of acetylcholinesterase against paraoxon - SAR study
Publication without faculty affiliation
publication
Evaluation of the Potency of Anti-HIV and Anti-HCV Drugs to Inhibit P-Glycoprotein Mediated Efflux of Digoxin in Caco-2 Cell Line and Human Precision-Cut Intestinal Slices
2022 |
Faculty of Pharmacy in Hradec Králové
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