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Molecular modelling
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PharmDr. Ondřej Holas Ph.D.
Academic staff at Faculty of Pharmacy in Hradec Králové
2 classes
53 publications
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class
Physical Principles of Dosage Forms
+1
GAPS308 |
Faculty of Pharmacy in Hradec Králové
Publications
publication
Monooxime bispyridinium reactivators bearing xylene linker synthesis and in vitro evaluation on model of organophosphate-inhibited acetylcholinesterase
2016 |
Faculty of Pharmacy in Hradec Králové
publication
Synthesis and in vitro evaluation of 7-methoxy-N-(pent-4-enyl)-1,2,3,4-tetrahydroacridin-9-amine - new tacrine derivate with cholinergic properties
2011 |
Faculty of Pharmacy in Hradec Králové, Faculty of Physical Education and Sport, First Faculty of Medicine
publication
Preparation, in vitro screening and molecular modelling of symmetrical 4-tert-butylpyridinium cholinesterase inhibitors - Analogues of SAD-128
2011 |
Faculty of Pharmacy in Hradec Králové
publication
Preparation, in vitro screening and molecular modelling of symmetrical bis-quinolinium cholinesterase inhibitors - implications for early Myasthenia gravis treatment
2011 |
Publication without faculty affiliation
publication
Monooxime-monocarbamoyl bispyridinium xylene-linked reactivators of acetylcholinesterase - synthesis, in vitro and toxicity evaluation, and docking studies
2010 |
Central Library of Charles University
publication
Pseudo-catalytic scavenging: Searching for a suitable reactivator of phosphorylated butyrylcholinesterase
2010 |
Central Library of Charles University
publication
Evaluation of the Potency of Anti-HIV and Anti-HCV Drugs to Inhibit P-Glycoprotein Mediated Efflux of Digoxin in Caco-2 Cell Line and Human Precision-Cut Intestinal Slices
2022 |
Faculty of Pharmacy in Hradec Králové
publication
The importance of the coating material type and amount in the preparation of liquisolid systems based on magnesium aluminometasilicate carrier
2021 |
Faculty of Pharmacy in Hradec Králové
publication
Oligonucleotide Delivery across the Caco-2 Monolayer: The Design and Evaluation of Self-Emulsifying Drug Delivery Systems (SEDDS)
2021 |
Faculty of Pharmacy in Hradec Králové
publication
PLGA Based Nanospheres as a Potent Macrophage-Specific Drug Delivery System
2021 |
Faculty of Pharmacy in Hradec Králové
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