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Analogues
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doc. PharmDr. Jan Zitko Ph.D.
Academic staff at Faculty of Pharmacy in Hradec Králové
6 classes
54 publications
Classes
class
Basics of Molecular Modelling of Drugs
+3
GAF316 |
Faculty of Pharmacy in Hradec Králové
class
Computer Aided Drug Design
+1
GDEFCH07 |
Faculty of Pharmacy in Hradec Králové
Publications
publication
Design, Synthesis and Evaluation of N-pyrazinylbenzamides as Potential Antimycobacterial Agents
2018 |
Faculty of Pharmacy in Hradec Králové
publication
Synthesis and antimycobacterial evaluation of N-substituted 5-chloropyrazine-2-carboxamides
2013 |
Faculty of Pharmacy in Hradec Králové
publication
Pyrazinecarboxylic acid derivatives with antimycobacterial activity
2012 |
Faculty of Pharmacy in Hradec Králové
publication
Antimycobacterial evaluation of pyrazinoic acid reversible derivatives
2011 |
Faculty of Pharmacy in Hradec Králové
publication
Synthesis and antimycobacterial properties of N-substituted 6-amino-5-cyanopyrazine-2-carboxamides
2011 |
Faculty of Pharmacy in Hradec Králové
publication
Development of new antituberculous active pyrazines evaluated in co-operation with TAACF program within a period of 15 years
2010 |
Faculty of Pharmacy in Hradec Králové
publication
Antimycobacterial pyridine carboxamides: From design to in vivo activity
2023 |
Faculty of Pharmacy in Hradec Králové
publication
Hybridization Approach Toward Novel Antituberculars: Design, Synthesis, and Biological Evaluation of Compounds Combining Pyrazinamide and 4-Aminosalicylic Acid
2023 |
Faculty of Pharmacy in Hradec Králové
publication
N-Pyrazinylhydroxybenzamides as biologically active compounds: a hit-expansion study and antimicrobial evaluation
2023 |
Faculty of Pharmacy in Hradec Králové
publication
Improving Antimicrobial Activity and Physico-Chemical Properties by Isosteric Replacement of 2-Aminothiazole with 2-Aminooxazole
2022 |
Faculty of Pharmacy in Hradec Králové, Faculty of Medicine in Hradec Králové
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