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doc. PharmDr. Jan Zitko Ph.D.
Academic staff at Faculty of Pharmacy in Hradec Králové
6 classes
54 publications
Classes
class
Basics of Molecular Modelling of Drugs
+3
GAF316 |
Faculty of Pharmacy in Hradec Králové
class
Computer Aided Drug Design
+1
GDEFCH07 |
Faculty of Pharmacy in Hradec Králové
Publications
publication
Inhibitors of aminoacyl-tRNA synthetases as antimycobacterial compounds: An up-to-date review
2021 |
Faculty of Pharmacy in Hradec Králové
publication
Towards Novel 3-Aminopyrazinamide-Based Prolyl-tRNA Synthetase Inhibitors: In Silico Modelling, Thermal Shift Assay and Structural Studies
2021 |
Faculty of Pharmacy in Hradec Králové
publication
Substituted N-(Pyrazin-2-yl)benzenesulfonamides; Synthesis, Anti-Infective Evaluation, Cytotoxicity, and In Silico Studies
2020 |
Faculty of Pharmacy in Hradec Králové
publication
Old Drugs and New Targets as an Outlook for the Treatment of Tuberculosis
2018 |
Faculty of Pharmacy in Hradec Králové
publication
Ureidopyrazine Derivatives: Synthesis and Biological Evaluation as Anti-Infectives and Abiotic Elicitors
2017 |
Faculty of Pharmacy in Hradec Králové, Faculty of Medicine in Hradec Králové, Central Library of Charles University
publication
Design, synthesis and anti-mycobacterial evaluation of some new N-phenylpyrazine-2-carboxamides
2016 |
Faculty of Pharmacy in Hradec Králové
publication
Enoyl acyl carrier protein reductase inhibitors: an updated patent review (2011-2015)
2016 |
Faculty of Pharmacy in Hradec Králové
publication
Pyrazine derivatives: a patent review (June 2012-present)
2015 |
Faculty of Pharmacy in Hradec Králové
publication
Synthesis and anti-infective evaluation of 5-amino-N-phenylpyrazine-2-carboxamides
2015 |
Faculty of Pharmacy in Hradec Králové
publication
Antimycobacterial pyridine carboxamides: From design to in vivo activity
2023 |
Faculty of Pharmacy in Hradec Králové
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