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doc. PharmDr. Jan Zitko Ph.D.
Academic staff at Faculty of Pharmacy in Hradec Králové
6 classes
54 publications
Classes
class
Basics of Molecular Modelling of Drugs
+3
GAF316 |
Faculty of Pharmacy in Hradec Králové
class
Computer Aided Drug Design
+1
GDEFCH07 |
Faculty of Pharmacy in Hradec Králové
Publications
publication
Improving Antimicrobial Activity and Physico-Chemical Properties by Isosteric Replacement of 2-Aminothiazole with 2-Aminooxazole
2022 |
Faculty of Pharmacy in Hradec Králové, Faculty of Medicine in Hradec Králové
publication
N-pyridinylbenzamides: an isosteric approach towards new antimycobacterial compounds
2021 |
Faculty of Pharmacy in Hradec Králové
publication
3-Substituted N-Benzylpyrazine-2-carboxamide Derivatives: Synthesis, Antimycobacterial and Antibacterial Evaluation
2017 |
Faculty of Pharmacy in Hradec Králové
publication
Synthesis and Antimicrobial Evaluation of 6-Alkylamino-N-phenylpyrazine-2-carboxamides
2015 |
Faculty of Pharmacy in Hradec Králové
publication
Indole-2-carboxamide derivatives: a patent evaluation of WO2015036412A1
2015 |
Faculty of Pharmacy in Hradec Králové
publication
Synthesis, Antimycobacterial Activity and In Vitro Cytotoxicity of 5-Chloro-N-phenylpyrazine-2-carboxamides
2013 |
Faculty of Pharmacy in Hradec Králové
publication
Substituted 2-(2-phenylhydrazinyl)pyrazine, process of its preparation, its use and pharmaceutical composition containing thereof
Publication without faculty affiliation
publication
Antimycobacterial pyridine carboxamides: From design to in vivo activity
2023 |
Faculty of Pharmacy in Hradec Králové
publication
Hybridization Approach Toward Novel Antituberculars: Design, Synthesis, and Biological Evaluation of Compounds Combining Pyrazinamide and 4-Aminosalicylic Acid
2023 |
Faculty of Pharmacy in Hradec Králové
publication
N-Pyrazinylhydroxybenzamides as biologically active compounds: a hit-expansion study and antimicrobial evaluation
2023 |
Faculty of Pharmacy in Hradec Králové
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