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doc. Mgr. et Mgr. Rafael Doležal Ph.D.
External academic staff at Central Library of Charles University
132 publications
Publications
publication
Preparation, In Vitro Screening and Molecular Modelling of Monoquaternary Compounds Related to the Selective Acetylcholinesterase Inhibitor BW284c51
2015 |
Publication without faculty affiliation
publication
Ligand-based 3D QSAR analysis of reactivation potency of mono- and bis-pyridinium aldoximes toward VX-inhibited rat acetylcholinesterase
2015 |
Publication without faculty affiliation
publication
7-MEOTA-donepezil like compounds as cholinesterase inhibitors: Synthesis, pharmacological evaluation, molecular modeling and QSAR studies
2014 |
Faculty of Pharmacy in Hradec Králové, Faculty of Science
publication
Comparison of Novel Tacrine and 7-MEOTA Derivatives with Aromatic and Alicyclic Residues: Synthesis, Biological Evaluation and Docking Studies
2013 |
First Faculty of Medicine, Faculty of Pharmacy in Hradec Králové
publication
Comparison of Novel Tacrine and 7-MEOTA Derivatives with Aromatic and Alicyclic Residues: Synthesis, Biological Evaluation and Docking Studies
2013 |
Faculty of Pharmacy in Hradec Králové
publication
Oximes: Inhibitors of Human Recombinant Acetylcholinesterase. A Structure-Activity Relationship (SAR) Study
+1
2013 |
Publication without faculty affiliation
publication
Quantitative structure-electrochemistry relationship of 1-phenyl-5-benzyl-sulfanyltetrazoles and their electrooxidation as a metabolic model
2010 |
Central Library of Charles University
publication
Graphic demonstration of the structure-antimycobacterial activity relationships in the series of ester phenylcarbamic acids with piperidine or pyrrolidine moiety
2008 |
Central Library of Charles University, Faculty of Pharmacy in Hradec Králové
publication
QSAR study of antimycobacterial activity of esters of substituted phenylcarbamic acids
2008 |
Central Library of Charles University, Faculty of Pharmacy in Hradec Králové
publication
The use of Toppliss approach to development of new antimycobacterial compounds: N-Benzylsalicylthioamides
2008 |
Central Library of Charles University, Faculty of Pharmacy in Hradec Králové
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