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c-h activation
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RNDr. Martin Novák Ph.D.
External academic staff at Faculty of Pharmacy in Hradec Králové
15 publications
Publications
publication
2,6-Disubstituted 7-(naphthalen-2-ylmethyl)-7H-purines as a new class of potent antitubercular agents inhibiting DprE1
2023 |
Faculty of Pharmacy in Hradec Králové
publication
Antimycobacterial pyridine carboxamides: From design to in vivo activity
2023 |
Faculty of Pharmacy in Hradec Králové
publication
Sustainable ionic liquids-based molecular platforms for designing acetylcholinesterase reactivators
2023 |
Faculty of Pharmacy in Hradec Králové
publication
Hybridization Approach Toward Novel Antituberculars: Design, Synthesis, and Biological Evaluation of Compounds Combining Pyrazinamide and 4-Aminosalicylic Acid
2023 |
Faculty of Pharmacy in Hradec Králové
publication
Structure-activity relationships of dually-acting acetylcholinesterase inhibitors derived from tacrine on N-methyl-D-Aspartate receptors
2021 |
Faculty of Pharmacy in Hradec Králové, Faculty of Science, Central Library of Charles University
publication
The Impact of Dextran Sodium Sulfate-Induced Gastrointestinal Injury on the Pharmacokinetic Parameters of Donepezil and Its Active Metabolite 6-O-desmethyldonepezil, and Gastric Myoelectric Activity in Experimental Pigs
2021 |
Faculty of Pharmacy in Hradec Králové, Faculty of Medicine in Hradec Králové
publication
Determination of Hypericin in Hypericum perforatum (St. John's Wort) Using Classical C18 and Pentafluorophenyl Stationary Phases: Contribution of Pi-Pi Interactions to High-Performance Liquid Chromatography (HPLC)
2019 |
Faculty of Pharmacy in Hradec Králové
publication
Synthesis, antimicrobial effect and lipophilicity-activity dependence of three series of dichained N-alkylammonium salts
2019 |
Publication without faculty affiliation
publication
Characterization of the penetration of the blood-brain barrier by high-performance liquid chromatography (HPLC) using a stationary phase with an immobilized artificial membrane
2018 |
Faculty of Education
publication
Phenoxytacrine derivatives: Low-toxicity neuroprotectants exerting affinity to ifenprodil-binding site and cholinesterase inhibition
2024 |
Faculty of Science, First Faculty of Medicine, Third Faculty of Medicine
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