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drug-resistance
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Ing. Vladimír Kubíček CSc.
Academic staff at Faculty of Pharmacy in Hradec Králové
56 publications
Publications
publication
Alkylamino derivatives of N-benzylpyrazine-2-carboxamide: synthesis and antimycobacterial evaluation
2015 |
Faculty of Pharmacy in Hradec Králové
publication
The metabolism of flubendazole and the activities of selected biotransformation enzymes in Haemonchus contortus strains susceptible and resistant to anthelmintics
2012 |
Faculty of Pharmacy in Hradec Králové
publication
Direct Amination of Nitroquinoline Derivatives via Nucleophilic Displacement of Aromatic Hydrogen
2021 |
Faculty of Pharmacy in Hradec Králové
publication
Substituted N-(Pyrazin-2-yl)benzenesulfonamides; Synthesis, Anti-Infective Evaluation, Cytotoxicity, and In Silico Studies
2020 |
Faculty of Pharmacy in Hradec Králové
publication
N-Pyrazinoyl Substituted Amino Acids as Potential Antimycobacterial Agents-the Synthesis and Biological Evaluation of Enantiomers
2020 |
Faculty of Pharmacy in Hradec Králové
publication
Carbonyl Reduction of Flubendazole in the Human Liver: Strict Stereospecificity, Sex Difference, Low Risk of Drug Interactions
2019 |
Faculty of Pharmacy in Hradec Králové, Faculty of Medicine in Hradec Králové
publication
Derivatives of 3-Aminopyrazine-2-carboxamides: Synthesis, Antimicrobial Evaluation, and in Vitro Cytotoxicity
2019 |
Faculty of Pharmacy in Hradec Králové
publication
Synthesis of Novel Pyrazinamide Derivatives Based on 3-Chloropyrazine-2-carboxamide and Their Antimicrobial Evaluation
2017 |
Faculty of Pharmacy in Hradec Králové
publication
The inhibitory effects of beta-caryophyllene, beta-caryophyllene oxide and alpha-humulene on the activities of the main drug-metabolizing enzymes in rat and human liver in vitro
2017 |
Faculty of Pharmacy in Hradec Králové
publication
Nerolidol and Farnesol Inhibit Some Cytochrome P450 Activities but Did Not Affect Other Xenobiotic-Metabolizing Enzymes in Rat and Human Hepatic Subcellular Fractions
2017 |
Faculty of Pharmacy in Hradec Králové
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