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doc. PharmDr. Jan Korábečný Ph.D.
External academic staff at Faculty of Pharmacy in Hradec Králové
179 publications
Publications
publication
Multi-target-directed therapeutic potential of 7-methoxytacrine-adamantylamine heterodimers in the Alzheimer's disease treatment
2017 |
Publication without faculty affiliation
publication
Inhibitors of Acetylcholinesterase Derived from 7-Methoxytacrine and Their Effects on the Choline Transporter CHT1
2017 |
Publication without faculty affiliation
publication
Synthesis, antimicrobial evaluation and molecular modeling of 5-hydroxyisoquinolinium salt series; the effect of the hydroxyl moiety
2016 |
Faculty of Pharmacy in Hradec Králové
publication
Towards understanding the mechanism of action of antibacterial N-alkyl-3-hydroxypyridinium salts: Biological activities, molecular modeling and QSAR studies
2016 |
Publication without faculty affiliation
publication
Ligand-based 3D QSAR analysis of reactivation potency of mono- and bis-pyridinium aldoximes toward VX-inhibited rat acetylcholinesterase
2015 |
Publication without faculty affiliation
publication
Variable Elimination Approaches for Data-Noise Reduction in 3D QSAR Calculations
2015 |
Publication without faculty affiliation
publication
Acetylcholinesterase inhibitors used or tested in Alzheimer’s disease therapy; their passive diffusion through blood brain barrier: In vitro study
2013 |
Publication without faculty affiliation
publication
Preparation of the pyridinium salts differing in the length of N-alkyl substituent
2010 |
Central Library of Charles University
publication
Phenoxytacrine derivatives: Low-toxicity neuroprotectants exerting affinity to ifenprodil-binding site and cholinesterase inhibition
2024 |
First Faculty of Medicine, Faculty of Science, Third Faculty of Medicine
publication
In silico library screening to find novel anticancer agent with chemosensitizing properties: focus on targeting ataxia telangiectasia and Rad3 related kinase
2024 |
Faculty of Medicine in Hradec Králové
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