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Mgr. Pavel Bárta Ph.D.
Akademický pracovník na Farmaceutická fakulta v Hradci Králové
31 publikací
Publikace
publication
Design, Synthesis and Antimicrobial Evaluation of New N-(1-Hydroxy-1,3-dihydrobenzo[c][1,2]oxaborol-6-yl)(hetero)aryl-2-carboxamides as Potential Inhibitors of Mycobacterial Leucyl-tRNA Synthetase
2023 |
Farmaceutická fakulta v Hradci Králové
publication
Design, synthesis and biological evaluation of substituted 3-amino-N-(thiazol-2-yl)pyrazine-2-carboxamides as inhibitors of mycobacterial methionine aminopeptidase 1
2022 |
Farmaceutická fakulta v Hradci Králové
publication
5-Alkylamino-N-phenylpyrazine-2-carboxamides: Design, Preparation, and Antimycobacterial Evaluation
2020 |
Farmaceutická fakulta v Hradci Králové
publication
Trans-resveratrol, but not other natural stilbenes occurring in food, carries the risk of drug-food interaction via inhibition of cytochrome P450 enzymes or interaction with xenosensor receptors
2019 |
Farmaceutická fakulta v Hradci Králové
publication
Entecavir Interacts with Influx Transporters hOAT1, hCNT2, hCNT3, but Not with hOCT2: The Potential for Renal Transporter-Mediated Cytotoxicity and Drug-Drug Interactions
2016 |
Farmaceutická fakulta v Hradci Králové
publication
The involvement of selected membrane transport mechanisms in the cellular uptake of Lu-177-labeled bombesin, somatostatin and gastrin analogues
2015 |
Farmaceutická fakulta v Hradci Králové
publication
Determination of receptor protein binding site specificity and relative binding strength using a time-resolved competition assay
2014 |
Farmaceutická fakulta v Hradci Králové
publication
Gefitinib Induces Epidermal Growth Factor Receptor Dimers Which Alters the Interaction Characteristics with (125)I-EGF
2011 |
Publikace bez příslušnosti k fakultě
publication
Insight into the Antibacterial Action of Iodinated Imine, an Analogue of Rafoxanide: a Comprehensive Study of Its Antistaphylococcal Activity
2023 |
Farmaceutická fakulta v Hradci Králové
publication
Antimycobacterial pyridine carboxamides: From design to in vivo activity
2023 |
Farmaceutická fakulta v Hradci Králové
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