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Mgr. Pavel Bárta Ph.D.
Academic staff at Faculty of Pharmacy in Hradec Králové
31 publications
Publications
publication
Hybridization Approach Toward Novel Antituberculars: Design, Synthesis, and Biological Evaluation of Compounds Combining Pyrazinamide and 4-Aminosalicylic Acid
2023 |
Faculty of Pharmacy in Hradec Králové
publication
Improving Antimicrobial Activity and Physico-Chemical Properties by Isosteric Replacement of 2-Aminothiazole with 2-Aminooxazole
2022 |
Faculty of Pharmacy in Hradec Králové, Faculty of Medicine in Hradec Králové
publication
Preparation, In Vitro Affinity, and In Vivo Biodistribution of Receptor-Specific 68Ga-Labeled Peptides Targeting Vascular Endothelial Growth Factor Receptors
2022 |
Faculty of Pharmacy in Hradec Králové
publication
Design, synthesis and biological evaluation of substituted 3-amino-N-(thiazol-2-yl)pyrazine-2-carboxamides as inhibitors of mycobacterial methionine aminopeptidase 1
2022 |
Faculty of Pharmacy in Hradec Králové
publication
Adenosine-Mimicking Derivatives of 3-Aminopyrazine-2-Carboxamide: Towards Inhibitors of Prolyl-tRNA Synthetase with Antimycobacterial Activity
2022 |
Faculty of Pharmacy in Hradec Králové
publication
Preclinical evaluation of anti-VEGFR2 monoclonal antibody ramucirumab labelled with zirconium-89 for tumour imaging
2021 |
Faculty of Pharmacy in Hradec Králové
publication
N-Pyrazinoyl Substituted Amino Acids as Potential Antimycobacterial Agents-the Synthesis and Biological Evaluation of Enantiomers
2020 |
Faculty of Pharmacy in Hradec Králové
publication
Antiangiogenic Human Monoclonal Antibody Ramucirumab Radiolabelling: In Vitro Evaluation on VEGFR2-positive Cell Lines
2019 |
Faculty of Pharmacy in Hradec Králové
publication
In vitro evaluation of concentration, labeling effectiveness and stability for I-131-labeled radioimmunoassay ligand using real-time detection technology
2017 |
Faculty of Pharmacy in Hradec Králové
publication
The effect of chelator type on in vitro receptor binding and stability in Lu-177-labeled cetuximab and panitumumab
2014 |
Faculty of Pharmacy in Hradec Králové
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