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Mgr. Pavel Bárta Ph.D.
Academic staff at Faculty of Pharmacy in Hradec Králové
31 publications
Publications
publication
Antimycobacterial pyridine carboxamides: From design to in vivo activity
2023 |
Faculty of Pharmacy in Hradec Králové
publication
Design, Synthesis and Antimicrobial Evaluation of New N-(1-Hydroxy-1,3-dihydrobenzo[c][1,2]oxaborol-6-yl)(hetero)aryl-2-carboxamides as Potential Inhibitors of Mycobacterial Leucyl-tRNA Synthetase
2023 |
Faculty of Pharmacy in Hradec Králové
publication
Hybridization Approach Toward Novel Antituberculars: Design, Synthesis, and Biological Evaluation of Compounds Combining Pyrazinamide and 4-Aminosalicylic Acid
2023 |
Faculty of Pharmacy in Hradec Králové
publication
Preparation, In Vitro Affinity, and In Vivo Biodistribution of Receptor-Specific 68Ga-Labeled Peptides Targeting Vascular Endothelial Growth Factor Receptors
2022 |
Faculty of Pharmacy in Hradec Králové
publication
Adenosine-Mimicking Derivatives of 3-Aminopyrazine-2-Carboxamide: Towards Inhibitors of Prolyl-tRNA Synthetase with Antimycobacterial Activity
2022 |
Faculty of Pharmacy in Hradec Králové
publication
Synthesis, Biological Evaluation, and In Silico Modeling of N-Substituted Quinoxaline-2-Carboxamides
2021 |
Faculty of Pharmacy in Hradec Králové
publication
Trans-resveratrol, but not other natural stilbenes occurring in food, carries the risk of drug-food interaction via inhibition of cytochrome P450 enzymes or interaction with xenosensor receptors
2019 |
Faculty of Pharmacy in Hradec Králové
publication
Antiangiogenic Human Monoclonal Antibody Ramucirumab Radiolabelling: In Vitro Evaluation on VEGFR2-positive Cell Lines
2019 |
Faculty of Pharmacy in Hradec Králové
publication
Entecavir Interacts with Influx Transporters hOAT1, hCNT2, hCNT3, but Not with hOCT2: The Potential for Renal Transporter-Mediated Cytotoxicity and Drug-Drug Interactions
2016 |
Faculty of Pharmacy in Hradec Králové
publication
The in vivo disposition and in vitro transmembrane transport of two model radiometabolites of DOTA-conjugated receptor-specific peptides labelled with Lu-177
2015 |
Faculty of Pharmacy in Hradec Králové
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