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IC50
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publication
Point and Interval Estimates of IC50
2011 |
Faculty of Medicine in Hradec Králové
publication
Point and Interval Estimates of IC50 by Line Approximation
2013 |
Faculty of Medicine in Hradec Králové
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Influence of some alkaloids from Eschscholtzia californica CHAM. (Papaveraceae) on human erythrocytic acetylcholinesterase: An screening study
Publication without faculty affiliation
publication
Influence of isoquinoline alkaloids from fraction A (chlorides soluble in chloroform) from Corydalis cava (Fumariaceae) on cholinesterases
Publication without faculty affiliation
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Comparison of the electronic properties, and thermodynamic and kinetic parameters of the aquation of selected platinum (II) derivatives with their anticancer IC50 indexes
2008 |
Faculty of Mathematics and Physics
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Cytotoxicity of acetylcholinesterase reactivators evaluated in vitro and its relation to their structure
2019 |
Publication without faculty affiliation
publication
Structure-activity relationship of quaternary acetylcholinesterase inhibitors - outlook for early Myasthenia gravis treatment
2010 |
Central Library of Charles University
publication
Susceptibility of clinical isolates of Leishmania aethiopica to miltefosine, paromomycin, amphotericin B and sodium stibogluconate using amastigote-macrophage in vitro model
2013 |
Faculty of Science
publication
Progress report of project realization "Morpholine inhibitors of DNA-dependent protein kinase as a potential radio-and chemosensitizing agent of tumor cells "
Publication without faculty affiliation
publication
DNA-proteinkinase inhibition; oncology treatment; chemosensitization
Publication without faculty affiliation
publication
Naturally occurring flavonoids as inhibitors of purified cytosolic glutathione S-transferase
2012 |
Faculty of Pharmacy in Hradec Králové
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Synthetic N-Acetyl-D-glucosamine Based Fully Branched Tetrasaccharide, a Mimetic of the Endogenous Ligand for CD69, Activates CD69 Killer Lymphocytes upon Dimerization via a Hydrophilic Flexible Linker
2010 |
Faculty of Science
publication
Substituted pyrazinecarboxamides: Synthesis and biological evaluation
2006 |
First Faculty of Medicine
publication
Design, Synthesis and in vitro Evaluation of Indolotacrine Analogues as Multitarget-Directed Ligands for the Treatment of Alzheimer's Disease
2016 |
Publication without faculty affiliation
publication
Discovery of multifunctional anti-Alzheimer's agents with a unique mechanism of action including inhibition of the enzyme butyrylcholinesterase and gamma-aminobutyric acid transporters
2021 |
Publication without faculty affiliation
publication
Isoquinoline alkaloids as prolyl oligopeptidase inhibitors
2015 |
Publication without faculty affiliation
publication
Privileged multi-target directed propargyl-tacrines combining cholinesterase and monoamine oxidase inhibition activities
2022 |
Faculty of Medicine in Hradec Králové
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Corylucinine, a new Alkaloid from Corydalis cava (Fumariaceae), and its Cholinesterase Activity
2012 |
Faculty of Pharmacy in Hradec Králové
publication
Enantiospecific effects of chiral drugs on cytochrome P450 inhibition in vitro
2016 |
Faculty of Pharmacy in Hradec Králové
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Proliferation inhibition of novel diphenylamine derivatives
2019 |
Publication without faculty affiliation
publication
Assessment of agonistic and antagonistic properties of widely used oral care antimicrobial substances toward steroid estrogenic and androgenic receptors
2019 |
Faculty of Science
publication
Inhibition of In Vitro Leukotriene B-4 Biosynthesis in Human Neutrophil Granulocytes and Docking Studies of Natural Quinones
2013 |
Faculty of Science
publication
Effect of Simvastatin, Coenzyme Q10, Resveratrol, Acetylcysteine and Acetylcarnitine on Mitochondrial Respiration
2016 |
First Faculty of Medicine
publication
Structure-Activity Relationships of N-benzylsalicylamides for Inhibition of Photosynthetic Electron Transport
2015 |
Faculty of Pharmacy in Hradec Králové
publication
Methylacridinium and its cholinergic properties
2009 |
Central Library of Charles University
publication
Methylacridinium and its cholinergic properties
2009 |
Central Library of Charles University, Faculty of Pharmacy in Hradec Králové
publication
Physicochemical and biological properties of novel amide-based steroidal inhibitors of NMDA receptors
2017 |
Central Library of Charles University, First Faculty of Medicine, Faculty of Mathematics and Physics
publication
Sugar modified pyrimido[4,5-b] indole nucleosides: synthesis and antiviral activity
2017 |
Faculty of Science
publication
Design, synthesis, and biological evaluation of 1-benzylamino-2-hydroxyalkyl derivatives as new potential disease-modifying multifunctional anti-Alzheimer's agents
2018 |
Publication without faculty affiliation
publication
New dual small molecules for Alzheimer's disease therapy combining histamine H-3 receptor (H3R) antagonism and calcium channels blockade with additional Cholinesterase inhibition
2019 |
Publication without faculty affiliation