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multitarget
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publication
Multitargeting nature of muscarinic orthosteric agonists and antagonists
2022 |
First Faculty of Medicine
publication
Phenothiazine-Tacrine Heterodimers: Pursuing Multitarget Directed Approach in Alzheimer's Disease
2021 |
Publication without faculty affiliation
publication
Novel multitarget-directed ligands aiming at symptoms and causes of Alzheimer's disease
2018 |
Publication without faculty affiliation
publication
Multitarget-Directed Ligands Combining Cholinesterase and Monoamine Oxidase Inhibition with Histamine H3R Antagonism for Neurodegenerative Diseases
2017 |
Publication without faculty affiliation
publication
Design, Synthesis and in vitro Evaluation of Indolotacrine Analogues as Multitarget-Directed Ligands for the Treatment of Alzheimer's Disease
2016 |
Publication without faculty affiliation
publication
Multitarget Drug Design Strategy: Quinone-Tacrine Hybrids Designed To Block Amyloid-beta Aggregation and To Exert Anticholinesterase and Antioxidant Effects
2014 |
Publication without faculty affiliation
publication
Novel 8-Hydroxyquinoline derivatives as multitarget compounds for the treatment of Alzheimer's disease
2016 |
Publication without faculty affiliation
publication
Crizotinib - multitargeted inhibitor in targeted NSCLC therapy
Publication without faculty affiliation
publication
Multitarget tacrine hybrids with neuroprotective properties to confront Alzheimer's disease
2017 |
Publication without faculty affiliation
publication
Bis-Amiridines as Acetylcholinesterase and Butyrylcholinesterase Inhibitors: N-Functionalization Determines the Multitarget Anti-Alzheimer's Activity Profile
2022 |
Publication without faculty affiliation
publication
Crizotinib - a multitargeted inhibitor as a molecularly targeted treatment in non small cell lung cancer
2013 |
Publication without faculty affiliation
publication
N-Alkyl-2-[4-(trifluoromethyl)benzoyl]hydrazine-1-carboxamides and Their Analogues: Synthesis and Multitarget Biological Activity
2020 |
Faculty of Pharmacy in Hradec Králové
publication
Amiridine-piperazine hybrids as cholinesterase inhibitors and potential multitarget agents for Alzheimer's disease treatment
2021 |
Publication without faculty affiliation
publication
Design and synthesis of novel tacrine-indole hybrids as potential multitarget-directed ligands for the treatment of Alzheimer's disease
2021 |
Publication without faculty affiliation
publication
Tacrine - Benzothiazoles: Novel class of potential multitarget anti-Alzheimer's drugs dealing with cholinergic, amyloid and mitochondrial systems
2021 |
Central Library of Charles University, Faculty of Medicine in Hradec Králové
publication
Synthesis and biological assessment of KojoTacrines as new agents for Alzheimer's disease therapy
2019 |
Publication without faculty affiliation
publication
Tacrine-resveratrol fused hybrids as multi-target-directed ligands against Alzheimer's disease
2017 |
Publication without faculty affiliation
publication
Physicochemistry shapes bioactivity landscape of pan-ABC transporter modulators: Anchor point for innovative Alzheimer's disease therapeutics
2022 |
Publication without faculty affiliation
publication
Effects of Novel Tacrine Derivatives on Mitochondrial Energy Metabolism and Monoamine Oxidase Activity-In Vitro Study
2021 |
First Faculty of Medicine
publication
Synthesis and biological evaluation of benzochromenopyrimidinones as cholinesterase inhibitors and potent antioxidant, non-hepatotoxic agents for Alzheimer's disease
2016 |
Publication without faculty affiliation
publication
Old Drugs and New Targets as an Outlook for the Treatment of Tuberculosis
2018 |
Faculty of Pharmacy in Hradec Králové
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Discovery of Dual A beta/Tau Inhibitors and Evaluation of Their Therapeutic Effect on a Drosophila Model of Alzheimer's Disease
2022 |
Publication without faculty affiliation
publication
Hydroxy-substituted trans-cinnamoyl derivatives as multifunctional tools in the context of Alzheimer's disease
2017 |
Publication without faculty affiliation
publication
Novel propargylamine-based inhibitors of cholinesterases and monoamine oxidases: Synthesis, biological evaluation and docking study
2021 |
Faculty of Pharmacy in Hradec Králové
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Cardanol-derived AChE inhibitors: Towards the development of dual binding derivatives for Alzheimer's disease
2016 |
Publication without faculty affiliation
publication
Regorafenib - the position of this drug in a current daily oncologic practice
2019 |
Publication without faculty affiliation
publication
Ladostigil - another pursuit of a dual action cognitive enhancer
2013 |
Publication without faculty affiliation
publication
A new look at 9-substituted acridines with various biological activities
2021 |
Publication without faculty affiliation
publication
Effect of Tapentadol on Experimental Model of Orofacial Pain - a Pilot Study
2020 |
First Faculty of Medicine, Third Faculty of Medicine
publication
(+/-)-BIGI-3h: Pentatarget-Directed Ligand combining Cholinesterase, Monoamine Oxidase, and Glycogen Synthase Kinase 3 beta Inhibition with Calcium Channel Antagonism and Antiaggregating Properties for Alzheimer's Disease
2021 |
Publication without faculty affiliation